Courbebaisse M, Quintrec ML, Zuber J, et al.
New Insight into Acute Effects of Cinacalcet on Calciuria in Kidney
Tranplanted Patients.
ASN Annual Meeting -- San Francisco
J Am Soc Nephrol
(Nov) 18:680A 2007

The calcimimetic Cinacalcet (CNC) decreases serum PTH and calcium (Ca)
concentrations in kidney transplanted patients with autonomous
hyperparathyroidism, but its acute effects on urinary Ca excretion has not
been reported. We studied the effect of CNC treatment in 23 kidney
transplanted patients. First, we compared serum PTH, total calcium (CaT),
phosphate (P) concentrations and GFR before and after CNC prescription
(chronic effect). Second, we analysed the kinetics of serum PTH, ionized
calcium (Cai) concentrations and urinary Ca excretion every hour during the
five hours following CNC morning dose (acute effect).
Chronic effect:
Morning fasting serum PTH decreased from 430.6
400.3 to 307.8
269.7 pg/ml (p =
0.005) and CaT from 2.82
0.24 to 2.54
0.21 mmol/l (p = 3.10-5), after 85
72 days of CNC treatment. Serum CaT-P ion product,
measured GFR (iohexol plasma clearance) and biochemical markers of bone
turnover were not modified by CNC treatment.
Acute effect: Serum PTH
levels fell within the hour following CNC dose, decreased by 51.5
20.7% 3 hours after treatment ingestion then
increased again. Serum Cai concentration decrease began 3 hours after CNC
ingestion and persisted beyond the fifth hour. Urinary Ca/ creatinine
excretion increased from the first hour, reached a maximum of 800
1139% then remained above the pretreatment values.
The analysis of the kinetics suggests that the decrease in Cai concentration
is mainly due to the marked increase in urinary Ca excretion. This is
supported by the normalization of Cai levels in 10 patients while serum PTH
concentrations remained elevated. The patients who normalized Cai
concentration after CNC administration had serum pre-treatment PTH values
below 240 pg/ml.
Conclusion: CNC treatment induced a transient and
marked increase in urinary Ca excretion that peaks 4 hours after treatment
intake. We suggest to check urinary Ca excretion at this time in order to
adapt water intake and prevent calcification
formation.
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