Rovin BH, McKinley A, Park EY, et al.
Oral Cyclophosphamide (POCY) in the Management of Severe Lupus
Glomerulonephritis (LN): An Under-Utilized Therapeutic Option.
ASN Annual Meeting -- San Diego
J Am Soc Nephrol
(Nov) 20:406A 2009

In our center, LN patients who do not enter a clinical trial are treated with
POCY for 2-4 months at a dose of 1.0-1.5 mg/kg ideal body weight. This
regimen uses about half the total dose of cyclophosphamide (CY) usually
reported in LN trials of POCY, and about the same amount of CY as the
standard 6 month course of intravenous CY (IVCY). After completing POCY
patients receive either azathioprine (AZA) or mycophenolate mofetil (MMF).
This regimen is well-tolerated and consistently associated with good
long-term outcomes. POCY is easy to administer and is less expensive than
IVCY as it is used in the United States. Here we report our experience with
POCY in 46 SLE patients with WHO class III, IV, and V LN treated between 1995
and 2006. Median follow-up was 23.5 months. Proteinuria improved or remained
stable in 90% of patients, and serum creatinine improved in 72% of patients
who had renal insufficiency at the initiation of therapy. Median time to
improvement was 5 months.
African Americans (AA) responded as well as
European Americans (EA) to treatment. Twelve months after initiation of
therapy 54% of AA and 60% of EA had achieved complete or partial remission.
Age, initial serum creatinine and initial level of proteinuria were not
different in patients that responded and those that did not. During follow-up
only 6 patients experienced new renal flares, and only 5 patients (11%) went
on to renal replacement therapy. Each patient who went to ESRD was poorly
compliant with medications. Adverse events resulted in discontinuation of
POCY in only 4 patients.
The main adverse events were leukopenia and
gastrointestinal upset, and each occurred in less than 10% of the cohort. One
patient developed amenorrhea, and no patients developed hemorrhagic cystitis.
In summary POCY followed by AZA or MMF is an effective sequential treatment
regimen for severe LN in both AA and EA, and has a favorable safety profile.
We therefore suggest that POCY remains a relevant treatment option for LN
that is easy to administer and less costly than IVCY.

© Copyright 2009-2010 American Society of
Nephrology.Reproduced with permission.
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