Bakris GL, Weir M, De Quattro V, Rosendorff C, McMahon G
Renal hemodynamic and antiproteinuric response to an ACE inhibitor (trandolapril) or calcium antagonist (verapamil) alone or in fixed dose combination in patients with diabetic nephropathy
Am Soc Nephrol
J Am Soc Nephrol (abstract) (Sep) 7:1546 1996

Proteinuria is a risk factor for subsequent progression of renal failure in many forms of renal disease and recent studies suggest ways in which various filtered proteins could exacerbate renal disease. In patients with type I and type II diabetic nephropathy, proteinuria is a hallmark of advanced structural disease and is a harbinger of progression in most cases.

Whereas ACE inhibitors have been shown to reduce proteinuria and protect renal function in diabetics, particularly those with type I nephropathy, the effects of calcium channel blockers on proteinuria have been more varied. Dihydropyridines such as nifedipine have been reported to increase proteinuria in some studies whereas verapamil and diltiazem have been reported to decrease proteinuria to a similar extent as ACE inhibitors.

In this study the authors examined the hypothesis that the fixed combination of the ACE inhibitor trandolapril with verapamil would reduce proteinuria in type II diabetics with nephropathy to a greater extent than either trandolapril or verapamil alone. They point out that these two agents have divergent effects on renal hemodynamics but that both can reduce proteinuria. Accordingly, they measured baseline renal hemodynamics, blood pressure and protein excretion rate in 39 type II diabetics with nephropathy then randomized the patients into three groups: 1) trandolapril; 2) verapamil and 3) trandolapril plus verapamil and measured GFR, RPF and proteinuria every 3 months for 12 months. Patients were maintained on a low sodium, low protein diet throughout the period of study. Baseline BP was elevated and baseline GFR and RPF were reduced.

They found that either drug alone or in combination normalized blood pressure (<140/90) but none of the regimens altered GFR or RPF significantly. In contrast, protein excretion was lowered about 40% in the single agent groups but by 70% in the combination of trandolapril plus verapamil, a difference that was significantly different compared to either drug alone. Furthermore, because the change in blood pressure from baseline and the and mean level after 12 months were not different between groups, the authors suggest that the anti-proteinuric effect of the fixed combination of trandolapril and verapamil may be due to changes in glomerular permeability.

Comment: The data from the study are provocative. The abstract does not supply information concerning the levels of dietary sodium and protein. Variability in these could influence differences observed in groups. It is also interesting that there were no detectable differences in GFR at 1 year in any group. Thus the divergent effects on renal hemodynamics between ACE inhibitors and verapamil claimed by the authors were not apparent at 1 year. Perhaps these occurred at 3 months then disappeared later (again data not presented). Still, this is an interesting finding and if confirmed would strengthen the argument for using the combination of an ACE inhibitor with a non-dihydropyridine calcium channel blocker in patients with type II diabetes. (Robert D. Toto, M.D., University of Texas Southwestern Medical Center)

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Am Soc Nephrol
H: Pathophysiology : Kidney in hypertension
CRF by problem area : Progression